Pharmacokinetic Studies on the Novel .BETA.2-Adrenoceptor Agonist TA-2005.
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چکیده
منابع مشابه
Indacaterol: a new once daily long-acting beta2 adrenoceptor agonist
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Beta(2)-adrenoceptor agonists such as fenoterol are anabolic in skeletal muscle, and because they promote hypertrophy and improve force-producing capacity, they have potential application for enhancing muscle repair after injury. No previous studies have measured the beta(2)-adrenoceptor population in regenerating skeletal muscle or determined whether fenoterol can improve functional recovery i...
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A fundamental question regarding receptor-G protein interaction is whether different agonists can lead a receptor to different intracellular signaling pathways. Our previous studies have demonstrated that although most beta(2)-adrenoceptor agonists activate both G(s) and G(i) proteins, fenoterol, a full agonist of beta(2)-adrenoceptor, selectively activates G(s) protein. Fenoterol contains two ...
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ژورنال
عنوان ژورنال: Drug Metabolism and Pharmacokinetics
سال: 1995
ISSN: 0916-1139
DOI: 10.2133/dmpk.10.497